5-Phenyl-1,3,4-oxadiazol-2(3H)-ones Are Potent Inhibitors of Notum Carboxylesterase Activity Identified by the Optimization of a Crystallographic Fragment Screening Hit
Mahy W., Willis NJ., Zhao Y., Woodward HL., Svensson F., Sipthorp J., Vecchia L., Ruza RR., Hillier J., Kjær S., Frew S., Monaghan A., Bictash M., Salinas PC., Whiting P., Vincent J-P., Jones EY., Fish PV.